Content
- Release form
- The composition of the drug Vinpotropil
- Pharmacological properties
- Pharmacodynamics and pharmacokinetics
- Indications for use
- Contraindications
- At what age can the drug be used?
- Instructions for use, dosage
- With VSD
- With osteochondrosis
- With dizziness
- Side effects
- Overdose
- special instructions
- Drug interactions
- Vinpotropil's analogs
- Piracesin
- Cereton
- Mexidol
- Terms, conditions of sale and storage
- Price
- Video about the drug Vinpotropil
Vinpotropil is a drug prescribed for various disorders and diseases of the brain. The drug has a wide range of indications, but requires extremely careful use.
Release form
The medicine is manufactured in Russia in the form of enteric capsules or tablets. The capsules are light yellow, the tablets are light brown with a grayish tint.
The product is contained in cell packs or polyethylene bottles and distributed in cardboard boxes.
The composition of the drug Vinpotropil
The medicine is made on the basis of 2 active components - pyrocetam and vinpocetine.
Additional composition:
- colloidal silicon dioxide;
- milk sugar;
- titanium dioxide;
- talc;
- gelatinous filler;
- dyes.
Pharmacological properties
The medication is a combined nootropic agent with vasodilating properties. The ingredients of the drug help to restore blood circulation in the brain and lower blood pressure. It also increases the resistance of brain cells to lack of oxygen, improves the transfer of oxygen and energy components to tissues.
The systematic intake of tablets leads to the accumulation of cAMP and ATP and an increase in the concentration of catecholamines. At the same time, the agent helps to relax the smooth muscles of the brain, enhances blood circulation in areas prone to ischemic attacks.
The drug causes a decrease in platelet aggregation, reduces blood viscosity and leads to deforming changes in red blood cells. Thanks to this action, the microcirculation in the brain is improved.
The drug helps to normalize metabolic processes, leads to an increase in the level of ATP in the brain tissues, improves the synthesis of RNA and phospholipids. In doing so, it helps to remove glucose components. The active substances of the agent normalize the cognitive functions of the brain, improve memory, and increase the ability to learn.
The drug allows you to get rid of violations displayed on the EEG, reduces the severity of vestibular disorders, improves synoptic communication, which leads to increased mental capacity and activity. In this case, the drug does not have a psychostimulating effect and does not cause drowsiness. The effect of the drug comes gradually.
Pharmacodynamics and pharmacokinetics
Vinpotropil (indications for the use of the agent are recommended to be studied in advance) has some pharmacokinetic and pharmacodynamic characteristics. The first active substance (vinpocetine) has good absorption capacity and is rapidly absorbed from the gastrointestinal tract. Bioavailability in this case is from 50 to 70%. The maximum concentration of the component in the blood is reached after 1 hour. Its half-life is about 5 hours.
Another main component (piracetam) enters the bloodstream of their gastrointestinal tract well and quickly. Bioavailability is about 95%. The maximum level of the ingredient in the blood is reached after 30-60 minutes. after taking. The substance is able to penetrate the BBB and has an accumulating ability. Its rate of excretion from cerebrospinal fluid is much lower than that of other tissues and systems.
The component does not lend itself to metabolic transformation. About 2/3 leaves the body unchanged through the renal system. Elimination rate - 30 min. The plasma half-life is approximately 4.5 hours. The substance is excreted from the brain within 7.5-8 hours.
Indications for use
The medicine is prescribed for various disorders of the brain, accompanied by impaired microcirculation or a decrease in cognitive functions.
Indications:
- impaired blood circulation in the brain (failure) due to previous strokes or encephalopathies of various origins;
- Parkinson's syndrome with a vascular etiology;
- toxic brain damage;
- brain injury;
- diseases of the nervous system, which are accompanied by a decrease in intellectual abilities;
- asthenic conditions;
- various forms of labyrinthopathy;
- organic psychosyndrome;
- kenotoses and migraines (as a preventive treatment).
Tablets / capsules should only be used as directed by a physician and after a diagnosis has been confirmed.
Contraindications
The drug has some limitations associated with the influence of active ingredients or special conditions of the patient's body.
Contraindications:
- arrhythmia (severe form of disorder);
- ischemic heart disease, occurring in a pronounced form;
- children under the age of 14;
- intolerance to the components;
- hemorrhagic stroke (acute course of pathology);
- hepatic and renal failure;
- pregnancy;
- lactation period.
Before taking the product, it is recommended to make sure that there are no allergic reactions to it.
At what age can the drug be used?
The medicine is approved for use in children over 14 years old. In this case, treatment should be carried out under the supervision of a specialist.
Instructions for use, dosage
Vinpotropil (indications for use contain an extensive list of diseases) is intended for oral use.
With VSD
With the development of vegetative-vascular dystonia (VVD), 1-2 capsules are prescribed 3 times a day. The duration of therapy can vary from several weeks to six months and is determined by the attending physician in each case separately. As a maintenance treatment, it is recommended to take 1 capsule 3 times a day.
With osteochondrosis
With osteochondrosis, the drug is taken according to the general scheme or according to the recommendations of a specialist. Course duration - individually from 2 weeks to 6 months.
With dizziness
With frequent dizziness, 1-2 capsules are prescribed 3 times a day. Duration of treatment - for several weeks or as recommended by a doctor.
Side effects
In most cases, the drug is well tolerated. In some cases, it can lead to the development of various reactions associated with the influence of active components or the individual characteristics of the patient's physiology.
Side effects:
- Disorders of the nervous system: increased excitability (mental or physical), impaired concentration, insomnia, anxiety, migraines, dizziness. Extrapyramidal disturbances, unbalanced behavior, irritability may also occur.
- Digestive dysfunctions: dyspeptic disorders, diarrhea or constipation, decreased appetite, various forms of gastralgia.
- Malfunctions of the cardiovascular system: worsening of the course of angina pectoris, increased heart rate, extrasystolic disturbances, decreased AV conduction rate.
- Other reactions: increased libido and sexual desire.
In the event of the listed signs, as well as symptoms not noted in the instructions, you should abandon the further use of the drug and consult a specialist for advice.
Overdose
There is no information on drug overdose. However, in case of exceeding daily or single doses and the development of any negative reactions, it is recommended to consult your doctor.
If necessary, symptomatic therapy is carried out - taking sorbents, washing the stomach, prescribing other medications.
special instructions
During the period of use of the drug, it is necessary to periodically undergo an ECG study. With long-term use of capsules / tablets, it is recommended to monitor kidney and liver function. Cancellation of the medication should be carried out gradually, systematically lowering the dosage.
The agent can have a negative effect on the central nervous system, therefore, it is recommended to exercise high caution. or refuse altogether to drive a car or carry out work that requires the speed of psychomotor reactions.
Drug interactions
Vinpotropil is capable of reacting with other drugs that have different or similar indications. Thus, the combined use of capsules / tablets with heparin increases the risks of developing hemorrhagic complications. The simultaneous appointment of a drug with thyroid hormones, antipsychotics and indirect anticoagulants can lead to an increase in the effectiveness of the second drugs.
A decrease in the therapeutic effect is observed with the combined use of the main agent with anticonvulsants. When using other medications during the period of administration of capsules / tablets, you should inform the treating person about this in advance. specialist, which will avoid the development of accidental interaction and, as a result, eliminate all risks of negative reactions.
Vinpotropil's analogs
The medication can lead to the development of intolerance reactions or other side effects, and therefore, it is recommended to replace it with another drug similar in indications and action.
It is not recommended to prescribe and use generics on your own, since the wrongly chosen remedy can lead to various complications and worsen the patient's condition. The selection of a similar tool should be dealt with by a specialist, taking into account all the characteristics of the patient's body.
Piracesin
This product is produced in the Republic of Belarus in the form of enteric capsules. The main ingredients are piracetam and cinnarizine. The drug belongs to the group of nootropics and helps to improve blood circulation in the brain and restore metabolic processes in it.
Indications:
- disorders of cerebral circulation due to various factors - stroke;
- toxic brain damage;
- various types of encephalopathy;
- organic psychosyndrome;
- head and brain trauma;
- asthenic conditions;
- various forms of labyrinthopathy;
- Meniere's disease;
- preventive treatment of migraines and kenotoses;
- disorders of the central nervous system, which are accompanied by a deterioration in intellectual and mnestic ability;
- intellectual lag in children.
Reception rules: 1-2 capsules 3 times a day. The duration of therapy is from 1 to 3 months. It is recommended to take 2-3 such courses per year. Dosage regimen (for children from 5 years old): 1-2 capsules 1-2 times a day. The duration of treatment is individual according to the doctor's recommendations.
Contraindications:
- allergy to medication;
- failure of the kidneys and liver;
- pregnancy;
- lactation period;
- children under 5 years of age.
Dispensing conditions - prescription. The cost of a medicine in commercial and state pharmacies in Russia is 220-250 rubles.
Cereton
Vinpotropil (indications for the use of capsules / tablets are recommended to be further clarified with the attending physician) must be replaced with other means, taking into account such factors as the tolerance of the components, the form and severity of the disorder, the patient's age, the presence contraindications.
Cereton is manufactured in Russia in the form of enteric capsules, the active ingredient of which is choline alfoscerate. The drug belongs to the group of nootoric drugs and is used for various disorders of the brain functions.
Recommendations for use:
- rehabilitation after suffering brain and head injuries;
- recovery from strokes;
- organic psychosyndrome, occurring against the background of degenerative changes;
- deterioration of cognitive functions, including various forms of encephalopathy and dementia;
- senile pseudomelancholia.
Dosage regimen (during rehabilitation after strokes): 0.8 g (in the morning) and 0.4 g (in the evening) for six months. Admission rules (for dementia): 1 capsule 3 times a day. It is recommended to take the product after meals. The duration of therapy is from 3 months to six months.
Restrictions on the appointment:
- drug intolerance;
- acute course of hemorrhagic stroke;
- pregnancy;
- lactation period;
- age under 18 (due to insufficient information about the effect of the product on children).
System - dispensing - by prescription. The cost of a medicine in pharmacies in Moscow and the Moscow region ranges from 215 to 1400 rubles. depending on the dosage.
Mexidol
Vinpotropil (indications for the use of similar drugs may differ) can be replaced by a drug such as Maxidol. This generic is also available in Russia in the form of tablets for oral use. The active substance is ethylmethylhydroxypyridine succinate. The drug exhibits high antioxidant properties and is prescribed for various conditions caused by dysfunction of the brain.
Application area:
- ischemic disorders (as part of complex treatment);
- toxic brain damage caused by taking antipsychotic drugs;
- VSD;
- acute circulatory disorders in the brain (consequences);
- head trauma;
- cognitive dysfunction due to the development of atherosclerosis;
- various forms of encephalopathy;
- neurosis-like disorders;
- anxiety;
- withdrawal symptoms caused by alcohol intake;
- asthenic diseases;
- stressful situations.
Dosing regimen: orally, 125-250 mg 3 times a day. The duration of therapy depends on the form and severity of the disorder and can vary from several days to six months.
Contraindications:
- functional disorders of the kidneys and liver, proceeding in an acute form;
- allergy to lactose, lactase deficiency, glucose-galactose malabsorption syndrome;
- childhood;
- pregnancy;
- lactation period;
- intolerance to the components.
The implementation mode is prescription. Prices for the drug in regional and regional pharmacies in Russia vary from 225 to 480 rubles.
Terms, conditions of sale and storage
Capsules / tablets should be stored in a dry, dark place at temperatures up to 25 0C. Expiration date - 24 months from the date of production. Do not use the product after the expiration date indicated on the package. The sales system is according to the recipe.
Price
The cost of a medicine may differ slightly from each other depending on the region of sale and the sales pharmacy representative. You can clarify the cost and purchase the drug at any pharmacy located in your place of residence.
Region and region of sale | Nominal volume (dosage) | Price |
Moscow, Moscow region | Tablets, 30 pcs. | 120-270 rub. |
St. Petersburg | Capsules, 5 mg + 400 mg | 120-730 rub. |
Saint Petersburg (suburbs) | Tablets, 10 mg + 800 mg | RUB 95-785 |
Leningrad region | Tablets, 30 pcs. | RUB 165-235 |
Novgorod region | Tablets, 30 pcs. | 140-230 rub. |
Before using Vinotropil, it is recommended to carefully study the instructions for use of the drug and familiarize yourself with the indications and contraindications. Additionally, you should consult your doctor.
Video about the drug Vinpotropil
Vinpotropil capsules instructions for use: