Sustanon 250 (Sustanon-250). Instructions for use, price, reviews

Sustanon 250 is a medicine used with a lack of male sex hormones. The drug requires strict adherence to instructions and supervision by the attending physician.

Release form

The medicine is produced in Ireland in the form of an oily solution for intramuscular administration. The solution is poured into ampoules packed in cardboard containers.

Chemical composition

The preparation contains several active ingredients (mixture of esters).

The main substances of testosterone:

• decanoate;
• propionate;
• isocapronate;
• phenylpropionate.

As additional components used: benzyl alcohol (phenylcarbinol) and oil made from peanuts.

Pharmacological properties

This ingredient is necessary for the full development of male sex hormones and secondary sex characteristics in men. In an adult man, the component performs a supportive function responsible for an erection, maintaining libido, general well-being and the functioning of the prostate organ.

Taking the medication leads to an increase in the level of male sex hormones and balancing of other hormones in the body. Treatment with the agent helps to eliminate various negative manifestations caused by a lack of testosterone. This normalizes weight, increases muscle volume and mass, and increases bone density.

Also, the use of medication leads to recovery and enhancement of sexual function. The solution causes a decrease in lipoprotein levels, an increase in hemoglobin and hematocrit. Injections do not cause disturbances in the production of liver enzymes, however, they can provoke the growth of the prostate gland. However, the functional capacity of the organ does not change.

In patients with diabetes mellitus, there is an increase in insulin sensitivity or a decrease in the concentration of sugar in the body. The use of the medication in transsexual women causes an increase in secondary sexual characteristics (in the male pattern).

Pharmacodynamics and pharmacokinetics

Sustanon 250 (instructions for use of the drug must be strictly followed by patients), when introduced into the body, is converted into testosterone (despite its multicomponent nature). The maximum concentration of the ingredient is observed after 1-2 days. Indicators return to their original rate after 3 weeks. Approximately 98% of the component interacts with globulins. The substance lends itself to metabolic reactions in the liver.

About 90% of the ingredient is excreted by the renal system. Approximately 6% leaves the body through the intestines along with bile.

Indications for use

The drug is used for androgen deficiency (hypogonadism). A solution is prescribed in the presence of pronounced signs and only after confirmation of the diagnosis by laboratory methods.

Contraindications

Injections have some restrictions on their use.

Contraindications:

• intolerance to the components;
• allergy to auxiliary ingredients;
• malignant lesion of the prostate gland;
• the presence of malignant tumors in the mammary gland.

  

The solution can be used with extreme caution in the following conditions:

• age over 65;
• chronic high blood pressure;
• various forms of thrombophilia;
• migraine;
• chronic lung diseases;
• severe course of liver failure;
• renal failure (chronic form);
• heart failure;
• ischemic disorders;
• diabetes;
• hypertrophic changes in the prostate gland (benign course of the disease);
• epileptic seizures;
• apnea;
• overweight.

In these conditions, it is recommended to choose a different therapy regimen.

At what age can the drug be used?

There is no information on the use of the product in childhood. In this connection, it is recommended to use the solution with extreme caution in boys during puberty.

Instructions for use

Sustanon 250 (instructions for use of the solution informs about the need for mandatory preliminary studies) is intended for intramuscular injection (deep into the buttock).

The therapy is selected individually. The standard dosage is 1 ampoule once every 3 weeks.

Patients over 65 years of age require dosage adjustment (calculated individually).

Side effects

The drug can lead to undesirable reactions from various systems and internal organs.

Side effects:

• Neoplasms of various forms: the formation of tumors in the area of ​​the prostate gland.
• Reproductive system and mammary glands: female breast development, impaired ejaculation, decreased sperm count, pathological erection (more than 4 hours).
• Disorders in the skeletal system, muscle and connective tissue: pain in the muscle area (myalgia).
• Skin: itchy elements, acne.
• Metabolism: weight gain, fluid retention in the body.
• Gastrointestinal tract: development of nausea.
• Liver and bile ducts: changes in hepatic function.
• Blood and lymph: Increased production of red blood cells by the bone marrow.
• The vascular system: an increase in blood pressure.
• Mental disorders: increased nervousness, depression, mood swings, changes in sexual desire.
• Changes in indicators during research: a decrease in the level of lipoproteins, an increase in prostate specific agent, an increase in hemoglobin, red blood cells and hematocrit.
• General reactions at the injection sites: itchy elements, redness, inflammation, pain syndrome.

In the event of the development of the listed signs, as well as other symptoms not specified in the instructions, it is recommended to stop further use of the medication and consult a doctor.

Overdose

The injections have extremely low toxicity. With the introduction of higher doses, the development of a pathological erection is possible.

With the development of such signs, therapy should be discontinued. After normalization of the condition, treatment is continued at lower dosages.

special instructions

Sustanon 250 must be used with extreme caution, since non-compliance with the rules and instructions for its use can provoke the development of severe and dangerous consequences for health. When an erection occurs, which is accompanied by pain, therapy must be discontinued. The entire period of treatment should be controlled by the level of the hormone in the body. In the first year of therapy, mandatory examinations are carried out once every 3 months, then - once a year.

It is also necessary to undergo periodic examination of the prostate gland in order to exclude the development of malignant neoplasms. Additionally, laboratory tests for hematocrit, hemoglobin, lipid profile and liver function tests should be performed.

Breast cancer patients require constant monitoring of blood calcium levels. With its increase, it is necessary to conduct appropriate therapy, and then continue treatment with the hormone. If sodium and water retention occurs in the body, further injections must be stopped. Requires constant monitoring of patients with high risks or bleeding disorders.

It is necessary to systematically monitor the condition of patients who have migraine pain or epileptic seizures. In boys of puberty, constant monitoring of the condition and development of sexual characteristics and functions should be carried out.

Elderly patients require constant observation and monitoring of the dynamics of treatment, since at this age, there are high risks of the formation of malignant tumors and prostatic hyperplasia glands. It is not recommended to use the drug as a sports performance enhancer, as such use can lead to serious health problems. The medication does not have a negative effect on the psychomotor functions of a person.

Drug interactions

Drugs that affect enzymes can lead to a decrease in the concentration of the main agent, so dosage adjustments may be required.

Drug groups and their interactions:

• Anticoagulants (oral forms) - enhancing their action, it may be necessary to adjust the dosage of these funds.
• Insulin and other hypoglycemic drugs - it is possible to increase glucose tolerance and decrease insulin dosages; blood sugar monitoring is required.
• Glucocorticosteroids and ACTH - possibly increased formation of puffiness; risk groups - a patient with liver and heart diseases.
• Medicines that stimulate the production of liver enzymes - a decrease in the level of the basic solution is possible; injection dosage adjustment may be required.
• Drugs that suppress liver enzymes - can lead to an increase in the concentration of the main agent; a reduction in the dosage of injections may be necessary.

Changes in laboratory values ​​may also be observed. Thus, the drug can lead to a decrease in the level of the T4 hormone. In this case, the concentration of T3 remains unchanged. At the same time, the drug does not adversely affect the functional ability of the thyroid gland.

Analogs

Sustanon 250 (instructions for the use of injections do not inform about the duration of therapy, since this feature must be established by a specialist) in in rare cases, it can lead to the development of allergic reactions, and therefore, it can be replaced by others similar in indication and action medicines.

Similar drugs should be used only with the permission of a specialist and under his close supervision.

Similar means are selected taking into account the physiological characteristics of the patient and the nature of the course of the disorder.

It is forbidden to independently and uncontrollably use substitutes, since such drugs can lead to serious health consequences.

Nebido

Generic is produced in Germany in the form of a solution required for intramuscular administration. The chemically active substance is testosterone undecanoate. The drug is used in the treatment of androgen deficiency and other conditions caused by the disease.

Other recommendations for appointment:

• anemic disorders (refractory form of the disorder);
• malignant tumors of the mammary glands;
• the formation of bleeding in the uterus (menopause);
• other disorders caused by menopause (combined treatment).

The dosage is determined individually, based on the area of ​​application of the injections and the patient's physiology.

Contraindications:

• allergy to the composition;
• pregnancy;
• lactation;
• malignant tumors of the prostate gland;
• nephrotic syndrome;
• cancers in the mammary glands (for men).

Terms of sale - prescription.

The price of the medicine starts from 5350 rubles.

Androgel

This substitute is produced in Belgium in the form of a gel for external use. The active ingredient is testosterone. The indication for the use of the drug is endogenous insufficiency (as replacement therapy). The daily dosage is up to 5 g once, preferably in the morning. The maximum daily allowance should not exceed 10 g. The duration of the course is individual.

Restrictions on the use of the gel:

• carcinomas, formed in the area of ​​the mammary glands;
• malignant lesion of the prostate gland;
• allergy to components

Age restrictions - not established or information is missing. It is used only on the recommendation of a specialist.

It is forbidden to use the medicine during pregnancy and breastfeeding, as it may affect the fetus.

The gel can be used with extreme caution in the following cases:

• the presence of malignant tumors;
• failure of the kidneys, liver and heart (severe forms of disorders);
• ischemic diseases;
• high blood pressure (chronic course of the disease);
• migraine;
• epileptic seizures.

Dispensing conditions - prescription.

The cost of the drug is from 2340 to 2500 rubles.

Omnadren 250

Sustanon (250 instructions for use of the medication informs about the need for constant monitoring with side of the attending physician) should be replaced with other similar means only in case of extreme necessity. The drug is a complete structural analogue of domestic production. A mixture of ester compounds (testosterone) is used as active ingredients.

Recommendations for the appointment:

• hypogonadism in men;
• delayed sexual development;
• conditions due to castration;
• violation in the development of male germ cells;
• erectile dysfunction caused by a lack of male sex hormones.

The drug can be used in women in the treatment of diseases. Caused by excess estrogen production. Application rules: 1 ampoule once a month. The duration of use is determined by the attending physician.

Contraindications:

• hypersensitivity to the composition of the product;
• nephrotic syndrome;
• period of pregnancy;
• breast-feeding;
• cancers that develop in the area of ​​the breast or prostate gland.

There are no age restrictions. A careful assessment of the condition is required before using the drug in boys during puberty. The way of implementation is prescription. The cost of injections varies from 760 to 800 rubles.

Terms, conditions of sale and storage

• Ampoules should be stored in a dark and dry place at a temperature of 8 to 30 ⁰C.
• Expiration date - 5 years from the date of issue.
• Do not use after the expiration date stated on the package.
• Dispensing method - by prescription.

Price

Prices for injections may vary depending on the region where they are sold. You can clarify the availability of the solution, as well as find out its cost at any pharmacy located at the place of residence.

Region / region	Dosage form / dosage	Cost, rub.)
Moscow, Moscow region	Solution, 250 mg (1 ml)	745-830
St. Petersburg	Solution, 250 mg (1 ml)	770-870
Saint Petersburg (suburbs)	Solution, 250 mg (1 ml)	755-840
Leningrad region	Solution, 250 mg (1 ml)	780-800
Novgorod region	Solution, 250 mg (1 ml)	765-820

Before using Sustanon 250, you must read the instructions for its use and consult a doctor. If necessary, it is additionally recommended to study the reviews of patients who have already used the drug.

Video about the drug Sustanon

Anabolic steroid Sustanon 250: